Is a
Patent attributes
Current Assignee
Patent Jurisdiction
Patent Number
Patent Inventor Names
Masazumi Yamaguchi0
Andrew Xian Chen0
John Fan0
Date of Patent
April 15, 2014
0Patent Application Number
131822180
Date Filed
July 13, 2011
0Patent Primary Examiner
Patent abstract
A solid dispersion comprising ((1S)-1-((((1S)-1-benzyl-2,3-dioxo-3-(cyclopropylamino)propyl)amino)carbonyl)-3-methylbutyl)carbamic acid 5-methoxy-3-oxapentyl ester made amorphous in the presence of a water-soluble cellulosic polymer has improved storage stability. The solid dispersion also has improved solubility for an improved bioavailability.
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