Is a
Patent attributes
Current Assignee
Patent Jurisdiction
Patent Number
Patent Inventor Names
Yasuhiro Tsukimi0
Toshio Kokubo0
Toshiya Moriwaki0
Tsutomu Masuda0
Hiroshi Fujishima0
Klaus Urbahns0
Masahiro Shiroo0
Masaomi Tajimi0
...
Date of Patent
May 8, 2012
0Patent Application Number
130524820
Date Filed
March 21, 2011
0Patent Primary Examiner
Patent abstract
This invention relates to tetrahydro-naphthalene derivatives and salts thereof which are useful as an active ingredient of pharmaceutical preparations. The tetrahydro-naphthalene derivatives of the present invention have excellent activity as VR1 antagonist and useful for the prophylaxis and treatment of diseases associated with VR1 activity, in particular for the treatment of urinary incontinence, overactive bladder, urge urinary incontinence, chronic pain, neuropathic pain, post-operative pain, rheumatoid arthritic pain, neuralgia, neuropathies, algesia, nerve injury, ischaemia, neurodegeneration, stroke, inflammatory disorders, asthma and COPD.
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